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Recent Publications

H index 61 as of May 2016

Citations in Each Year
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2016

305     Heterogeneous Phase Transfer Catalysis in Solid Phase Syntheses of Anth-Cyclic Tetrapeptides, D. Xin, K.-Y. Wong, K. Burgess, J. Org. Chem., 2016, submitted.

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304     Small Molecules for Active Targeting in Cancer, C. S. Kue, A. Kamkaew, K. Burgess, L. V. Kiew, L. Y. Chung, H. B. Lee, Med. Res. Rev., 2016, 36, 494-575. DOI:10.1002/med.21387

303     Anthranilic Acid-containing Cyclic Tetrapeptides:  At the Crossroads of Conformational Rigidity and Synthetic Accessibility, D. Xin, K. Burgess, Org. Biomol. Chem., 2016, 14, 5049-5058. DOI: 10.1039/C6OB00693K

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302     Chitosan-coated poly(lactic-co-glycolic acid)-diiodinated boron-dipyrromethene nanoparticles improve tumor selectivity and stealth properties in photodynamic cancer therapy , L. Chung, K. Burgess, J. Mat. Chem. B, 2016, 12, 1431-1452. DOI:10.1166/jbn.2016.2263

2015

301       Aza-BODIPY Dyes With Enhanced Hydrophilicity, A. Kamkaew, K. Burgess, Chem. Comm., 2015, 51, 10664-7. DOI: 10.1039/C5CC03649F

300        Oligoethylene Glycol-substituted Aza-BODIPY Dyes as Red Emitting ER-Probes, S. Thavornpradit, T. Puangsamlee, A. Kamkaew, D. Xin, N. Wanichacheva, K. Burgess, Org. Biomol. Chem., 2015, 8271-6.  DOI:10.1039/c50b01104c

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299         Extended Piperidine-piperidinone Protein Interface Mimics, D. Xin, A. Raghuraman, K. Burgess, J. Org. Chem., 2015, 80, 4450-4458. (DOI:10.1021/acs.joc.5b00300

298         Protein-protein Interface Mimicry By An Oxazoline Piperidine-2,4-dione, X. Li, J. Taechalertpaisarn, D. Xin, K. Burgess, Org. Lett., 2015, 17, 632-635.  DOI:10.1021/ol5036547

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297         Targeted PDT Agent Eradicates TrkC Expressing Tumors Via Photodynamic Therapy (PDT), C. S. Kue, A. Kamkaew, H. B. Lee, L. Y. Chung, L. V. Kiew, K. Burgess, Mol. Pharmaceutics, 2015, 12, 212-22. DOI:1021/mp5005564

2014

296         In Vivo Studies of Nanostructure-Based Photosensitizers for Photodynamic Cancer Therapy, S. H. Voon, L. V. Kiew, H. B. Lee, S. H. Lim, M. I. Noordin, A. Kamkaew, K. Burgess and L. Y. Chung, Small, 2014, 10, 4993-5013. DOI:10.1002/smll.201401416

295         Small Molecule Probes that Perturb A Protein-protein Interface In Antithrombin, D. Xin, A. Holzenburg, K. Burgess, Chem. Sci., 2014, 5, 4914-4921. DOI:10.1039/c4sc01295j

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294         A Chemoselective Route to b-Enamino Esters and Thioesters, D. Xin, K. Burgess, Org. Lett., 2014, 16, 2108-2110.  DOI:10.1021/ol5005643

293         A Multi-faced Secondary Structure Mimics Based on Piperidine-Piperidinones, D. Xin, L. M. Perez, T. R. Ioerger, K. Burgess, Angew. Chem., Int. Ed., 2014, 53, 3594-3498. DOI:10.1002/anie.201400927

292         Metathesis for Catalyst Design:  Metacatalysis, S. Khumsubdee, K. Burgess, Tetrahedron, 2014, 70, 1326-35.

291         Rosamines Targeting the Cancer Oxidative Phosphorylation Pathway, S. H. Lim, L. Wu, V. Kiew, L. Y. Chung, K. Burgess, H. B. Lee, PLOS One, 2014, 9, e82934. DOI:10.1371/journal.pone.0082934

2013

290         Homo-Roche Ester Derivatives By Asymmetric Hydrogenation and Organocatalysis, S. Khumsubdee, H. Zhou, K. Burgess, J. Org. Chem., 2013, 78, 11948-55. DOI:10.1021/jo401996m

289         Double-targeting Using a TrkC-Ligand Conjugated to BODIPY-based PDT Agent, A. Kamkaew, K. Burgess, J. Med. Chem., 2013, 56, 7608-14. DOI:10.1021/jm4012142

288         A Comparison Between Oxazoline-imidazolinylidene, -imidazoylidine, -benzimidazoylidine Hydrogenations Catalysts, S. Khumsubdee, Y. Fan, K. Burgess, J. Org. Chem., 2013, 78, 9969-74. DOI:10.1021/jo4013783

287         Expanding the Scope of Oligo-pyrrolinone-pyrrolidines as Protein-protein Interface Mimics, A. Raghuraman, D. Xin, L. M. Perez, K. Burgess, J. Org. Chem., 2013, 78, 4823-4833. DOI:10.21/jo400323k

286         Evaluating Minimalist Mimics by Exploring Key Orientations on Secondary Structures (EKOS), D. Xin, E. Ko, L. M. Perez, T. R. Ioerger, K. Burgess, Org. Biomol. Chem. 2013, 11, 7789-801. DOI:10.1039/c3ob4184k

285     Comparison of Asymmetric Hydrogenations of Unsaturated-Carboxylic Acids and -Esters, S, Khumsubdee, K. Burgess, ACS Catalysis, 2013, 3, 237-249.

284     Highly Stereoselective Syntheses of all 1,2,3-Me,OH,Me Triads via Asymmetric Hydrogenation Reactions, Y. Zhu and K. Burgess, Adv. Synth. Cat., 2013, 355, 107-115. DOI:10.1002/adsc.201200709

283         Exploring Key Orientations at Protein-Protein Interfaces with Small Molecule Probes, E. Ko, A. Raghuraman, L. M. Perez, T. R. Ioerger, K. Burgess, J. Am. Chem. Soc., 2013, 135, 167-173.  DOI:10.1021/ja3067258

2012

282     Small Molecule Ligands for Active Targeting of TrkC-expressing Tumor Cells, E. Ko, A. Kamkaew, K. Burgess, ACS Med. Chem. Lett., 2012, 3, 1008-1012. DOI:10.1021/ml300227d

281     BODIPY Dyes in Photodynamic Therapy, A. Kamkaew, S. H. Lim, H. B. Lee, L. V. Kiew, L. Y. Chung, K. Burgess, Chem. Soc. Rev., 2012, 42, 77-88.  DOI:10.1039/c2cs3521h

280     Omegatides:  Constrained Analogs of Peptide Primary Sequence, D. Fedoseyenko, A. Raghuraman, E. Ko, K. Burgess, Org. Biomol. Chem., 2012, 10, 921-4. DOI:10.1039/c20b06692k

279     Iridium Catalyzed Enantioselective Hydrogenation of a-Alkoxy and b-Alkoxy Vinyl Ethers, Y. Zhu and K. Burgess, RSC Adv., 2012, 2, 4728-35. DOI:10.1039/c2ra01350a

278     Filling Gaps in Asymmetric Hydrogenation Methods for Acyclic Stereocontrol:  Application to Chirons for Polyketide-derived Natural Products, Y. Zhu and K. Burgess, Acct. Chem. Res., 2012, 45, 1623-36.  DOI:10.1021/ar200145q

277      (n4-1,5-Cyclooctadiene)(1-[(4S)-(2-(1-adamantyl)-4-5-dihydrooxazolyl)-ethyl]-3-(2,6-diisopropylphenyl)imidazolin-2-ylidene)iridium(I) Tetrakis(3,5-bis(tribluoromethyl)phenyl)borate, Y. Zhu, K. Burgess, EROS USGS, 2012.

2011

276 Continuous Flow Biocatalytic Resolutions of Methyl Sulfinylacetates, Z. Liu, K. Burgess, Tetrahedron Lett., 2011, 52, 6325-27.  DOI:10.1016/j.tetlet.2011.09.024

275     Asymmetric Syntheses of alpha-Methyl gamma-amino Acid Derivatives, Y. Zhu, S. Khumsubdee, A. Schaefer, K. Burgess, J. Org. Chem., 2011, 76, 7449-57. DOI:10.1021/jo201215c

274     Cationic Polyfluorenes for Intracellular Delivery of Proteins, A. Kamkaew, R. Barhoumi, R. C. Burghardt, K. Burgess, Org. Biomol. Chem., 2011, 9, 6513-8.  DOI:10.1039/c1ob05874f

273     Highly Efficient and Photostable Photonic Materials from Diiodinated BODIPY Laser Dyes, M. E. Pérez-Ojeda, C. Thivierge, V. Martin, A. Costela, K. Burgess and In. García-Moreno, Opt. Mat. Exp., 2011, 1, 243-51.

272     Pyrrolinone-pyrrolidine Oligomers as Universal Peptidomimetics, A. Raghuraman, E. Ko, K. Burgess, J. Am. Chem. Soc., 2011, 133, 12350-12351.  DOI:10.1021/ja2033734

271      Minimalist and Universal Peptidomimetics, E. Ko, J. Liu, K. Burgess, Chem. Soc. Rev., 2011, 40, 4411-4421.  DOI:10.1039/c0cs00218f

270     Brilliant BODIPY-fluorene Copolymers With Dispersed Absorption and Emission Maxima, C. Thivierge, A. Loudet, K. Burgess, Macromolecules, 2011, 44, 4012-4015. DOI:10.1021/ma200174w

269     Pyrrole-based Scaffolds for Turn Mimics, E. Ko, K. Burgess, Org. Lett., 2011, 13, 980-3. DOI:10.1021/ol103022m

268     Energy Transfer Cassettes in Silica Nanoparticles Target Intracellular Organelles, J. Jose, A. Loudet, Y. Ueno, L. Wu, H.-Y. Chen, D. H. Son, R. Barhoumi, R. Burghardt, K. Burgess, Org. Biomol. Chem., 2011, 9, 3871-77.

267     Universal Peptidomimetics, E. Ko, J. Liu, L.M. Perez, G. Lu, A. Schaefer, K. Burgess, J. Am. Chem. Soc., 2011, 133, 462-77.

266     Fluorescent Proton Sensors Based on Energy Transfer, C. Thivierge, J. Han, R. M. Jenkins, K. Burgess, J. Org. Chem., 2011, 76, 5219-28.

265     Organelle-selective Energy Transfer: A Fluorescent Indicator of Intracellular Environment, A. Loudet, Y. Ueno, L. Wu, J. Jose, R. Barhoumi, K. Burgess, Bioorg. Med. Chem. Lett., 2011, 21, 1849-51.

264     Encapsulated Energy Transfer Cassettes With Extremely Well Resolved Fluorescent Outputs, Y. Ueno, J. Jose, A. Loudet, C. Perez-Bolivar, P. Anzenbacher, K. Burgess, J. Am. Chem. Soc., 2011, 133, 51-5. PMID 21105708

2010

263     In Glaucoma the Up-regulated Truncated TrkC.T1 Receptor Isoform in Glia Causes Increased TNF-α Production, leading to retinal ganglion cell death, Y. Bai, Z. Shi, Y. Zhuo, J. Liu, A. Malakhov, E. Ko, K. Burgess, H. Schaefer, P. Esteban, L. Tessarollo, and H. Saragovi, Invest. Ophthal. Vis. Sci., 2010, 51, 6639-51.

262     Encapsulated Energy Transfer Cassettes With Extremely Well Resolved Fluorescent Outputs, Y. Ueno, J. Jose, A. Loudet, C. Perez-Bolivar, P. Anzenbacher, K. Burgess, J. Am. Chem. Soc., 2010, 133, 51-55.

261     An Asymmetric Hydrogenation Route To (-)-Spongidepsin, Y. Zhu, A. Loudet, K. Burgess, Org. Lett., 2010, 12, 4392-4395.

260     Bivalent Diketopiperazine-based TrkC Antagonists, J. Liu, F. Brahimi, H. U. Saragovi, K. Burgess, J. Med. Chem., 2010, 53, 5044-8.

259     A Monovalent Agonist of TrkA Tyrosine Kinase Receptors Can Be Converted into a Bivalent Antagonist, F. Brahimi, J. Liu, A. Malakhov, S. Chowdhury, E. Purisima, L. Ivanisevic, A. Caron, K. Burgess, H. Saragovi, Biochim. Biophys. Acta, 2010, 1800, 1018-26.

258     Intracellular imaging of organelles with new water-soluble benzophenoxazine dyes, J. Jose, A. Loudet, Y. Ueno, R. Barhoumi, R. C. Burghardt, K. Burgess, Org. Biomol. Chem., 2010, 8, 2052-9.

257    Carbene-metal-hydrides Can Be Much Less Acidic Than Phosphine-metal-hydrides: Significance in Hydrogenations, Y. Zhu, Y. Fan, K. Burgess, J. Am. Chem. Soc., 2010, 132, 6249-53.

256     A Combinatorial Approach for Targeted Delivery using Small Molecules and Reversible Masking to Bypass Non-Specific Uptake In Vivo, Q. Shi, A. Nguyen, Y. Angell, D. Deng, C.-R. Na, K. Burgess, D. Roberts, C. Brunicardi, N. Templeton, Gene Therapy, 2010, 17, 1085-97.

255     Fluorescent Indicators for Intracellular pH Ex Vivo, J. Han, K. Burgess, Chem. Rev., 2010, 110, 2709-28.

254     In Vitro and In Vivo Photo-cytotoxicity of Boron Dipyrromethene Derivatives for Photodynamic Therapy, S. H. Lim, C. Thivierge, P. Nowak-Sliwinska, J. Han, H. Van den Bergh, G. Wagnieres, K. Burgess, H. B. Lee, J. Med. Chem., 2010, 53, 2865-74.

2009

253     A Peptidomimetic of NT-3 acts as a TrkC antagonist, F. Brahimi, A. Malakhov, H. B. Lee, M. Pattawarapan, L. Ivanisevic, K. Burgess, H. U. Saragovi, Peptides, 2009, 1833-9.

252     Energy transfer dyads based on Nile Red, J. Jose, Y. Ueno, J.C. Castro, L. Li, K. Burgess, Tetrahedron Lett., 2009, 50, 6442-5.

251     Synthesis of Vicinal Dimethyl Chirons by Asymmetric Hydrogenation of Trisubstituted Alkenes, J. Zhao, K. Burgess, J. Am. Chem. Soc., 2009, 131, 13236-7.

250     New Cytotoxic Rosamine Derivatives Selectively Accumulate in the Mitochondria of Cancer Cells, S.A. Lim, L. Wu, K. Burgess, H.B. Lee, Anti-Cancer Drugs, 2009, 20, 461-8.

249     Fluorescent Cassettes for Monitoring Three-component Interactions In Vitro and Ex Vivo, L. Wu, A. Loudet, R. Barhoumi, R.C. Burghardt, K. Burgess, J. Am. Chem. Soc., 2009, 131, 9156-7.

248     Bivalent Peptidomimetic Ligands of TrkC are Biased Agonists, Selectively Induce Neuritogenesis, or Potentiate Neurotrophin-3 Trophic Signals, D. Chen, F. Brahimi, Y. Angell, Y.-C. Li, J. Moscowitz, H. U. Saragovi, K. Burgess, ACS Chem. Biol., 2009, 4, 769-81.

247     Synthesis of Regiosomerically Pure 5-Functionalized 2’, 7’–Dichlorofloresceins, K. Burgess, J. C. Castro, A. Malakhov, Synthesis, 2009, 7, 1224-6.

246    Aldol-type Chirons From Asymmetric Hydrogenations of Trisubstituted Alkenes, K. Burgess, J. Zhao, Org. Lett.,  2009, 11, 2053-6.

245     Photophysics and Stability of Cyano-Substituted Boradiazaindacene Dyes, K. Cieslik-Boczula, K. Burgess, L. Li, B. Nguyen, L. Pandey, W. M. De Borggraee, M. Van der Auweraer,  N. Boens, Physical Chem. Chem. Phys., 2009, 8, 1006-15.

244     A Ratiometric pH Reporter For Imaging Protein-dye Conjugates in Living Cells, J. Han, A. Loudet, R. Barhoumi, R. Burghardt, K. Burgess, J. Am. Chem. Soc., 2009, 131, 1642-3. 

243     Water-soluble Nile Blue Derivatives: Syntheses and Photophysical Properties, J. Jose, Y. Ueno, K. Burgess, Chem.—Eur. J., 2009, 15, 418-23.

242     3- and 5-Functionalized BODIPYs via The Liebeskind-Srogl Reaction, J. Han, O. Gonzalez, A. Aguilar-Aguilar, E. Pena-Cabrera K. Burgess, Org. Biomol. Chem., 2009, 7, 34-6.

2008

241     B,O-Chelated Azadipyrromethenes as Near-IR Probes, K. Burgess, A. Loudet, R. Bandichhor, A. Palma, S. McDonnell, M. Hall, Org. Lett., 2008, 10, 4771-4. (Highlighted in Synfacts 2009, 2, 150).

240     A New Synthesis of Symmetric Boraindacene (BODIPY) Dyes, L. Wu, K. Burgess, Chem. Commun., 2008, 40, 4933-5. 

239     Non-Covalent Delivery of Proteins into Mammalian Cells, A. Loudet, J. Han, R. Barhoumi, J-P. Pellois, R. C. Burghardt, K. Burgess, Org. Biomol. Chem., 2008, 6, 4516-22. 

238     Synthesis and Spectroscopic Properties of Rosamines with Cyclic Amine Substituents, L. Wu, K. Burgess, J. Org. Chem., 2008, 73, 8711-8.

237     Asymmetric Hydrogenation Approaches to Valuable, Acyclic 1,3-Hydroxymethyl Chirons, K. Burgess, Y. Zhu, J. Am. Chem. Soc., 2008, 130, 8894-5.  (Highlighted in Synfacts 2008, 11, 1176.)

236     Fluorescent Amino-and Thiopyronin Dyes, L. Wu, K. Burgess, Org. Lett., 2008, 10, 1779-82.  (Highlighted in Synfacts, 2008, 7, 699.)

235     Syntheses of Highly Fluorescent GFP-chromophore Analogs, L. Wu, K. Burgess, J. Am. Chem. Soc., 2008, 130, 4089-96.

234     Functionalization of the 4,4-Difluoro-4-bora-3a,4a-diaza-s-indacene (BODIPY) Core, L. Li, B. Nguyen, K. Burgess, Biorg. Med. Chem. Lett., 2008, 18, 3112-6.

233     Syntheses and Spectral Properties of Functionalized, Water-soluble BODIPY Derivatives, L. Li, J. Han, B. Nguyen, K. Burgess, J. Org. Chem., 2008, 73, 1963-70.

232     Iridium-Catalyzed Asymmetric Hydrogenation of Vinyl Ether, Y. Zhu, K. Burgess, Adv. Synth. Catal., 2008, 350, 979-83. (Highlighted in Synfacts 2008, 7, 733.)

231     Lipid Diffusion from Single Molecules of a Labeled Protein Undergoing Dynamic Association with Giant Unilamellar Vesicles and Supported Bilayers,  A. Sharonov, R. Bandichhor, K. Burgess, A. Petrescu, F. Schroeder, A. Kier, R. Hochstrasser, Langmuir, 2008, 24, 844-50. 

230     Functionalized BF2 Chelated Azadipyrromethene Dyes, A. Loudet, R. Bandichhor, L. Wu, K. Burgess, Tetrahedron, 2008, 64, 3642-54.

229     A Combinatorial Method for Solution-phase Synthesis of Labeled Bivalent β-Turn Mimics, Y. Angell, D. Chen, F. Brahimi, H. U. Saragovi, K. Burgess, J. Am. Chem. Soc., 2008, 130, 556-65.

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